99% Tianeptine sodium nnu CAS 30123-17-2
Nkọwapụta
ITEM | Ọkọlọtọ | Nsonaazụ |
Ọdịdị | Ọcha ka ntụ ntụ na-acha odo odo | White crystalline ntụ ntụ |
Solubility | Freely soluble Na mmiri na methanol na dichloromethane | Na-akwado |
njirimara | Site na IR, Dakọtara na ọkọlọtọ ọrụ | Na-akwado |
(2) Ọ na-enye mmeghachi omume nke sodium | Na-akwado | |
Ihe ndị na-adịghị ọcha A | ≤0.1% | Achọpụtaghị |
Ngwakọta ndị emetụtara | Otu adịghị ọcha ọ bụla kacha ≤0.1% | 0.060% |
Mkpokọta adịghị ọcha≤0.4% | 0.36% | |
Ihe mgbaze fọdụrụ (GC) | Acetidin ≤ 0.5% | ND |
Dichloromethane ≤ 0.06% | ND | |
Methanol ≤ 0.3% | ND | |
Acetone bụ 0.5% | 0.29% | |
Acetonitrile ≤0.041% | 0.022% | |
Ethanol ≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Mmiri | ≤5.0% | 3.8% |
Nyocha (HPLC) | 99.0% -101.0% (na anhydrousbasis) | 99.70% |
Ngwa
Tianeptine sodiumnnubụ tricyclic antidepressant.Usoro mgbochi ịda mbà n'obi dị iche na nke ndị antidepressants tricyclic ọdịnala.Ọ nwere ike iwelie iweghachite 5-HT na mgbawa synapti.Mmetụta nke HT neuronal conduction.Enweghị njikọ maka choline ma ọ bụ adrenergic receptors.Mmetụta antidepressant dị ka nke tricyclics, mana nnabata dị mma karịa nke tricyclics.Maka ọgwụgwọ nke ịda mbà n'obi dị nro ma ọ bụ nke siri ike, neurogenic na ịda mbà n'obi na-emeghachi omume, nchekasị na ịda mbà n'obi na anụ ahụ, karịsịa ahụ erughị ala nke eriri afọ, na nchekasị na ịda mbà n'obi na ndị ọrịa na-aṅụ mmanya na-aba n'anya n'oge nkwụsị.